

HY-16986A · 5 mg
MedChemExpress · Cat: HY-16986A
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medchemexpress.com/EPZ011989-trifluoroacetate.htmlDescription
EPZ-011989 trifluoroacetate is a potent and orally active Zeste Homolog 2 EZH2 inhibitor with metabolic stability. EPZ-011989 trifluoroacetate has inhibitory inhibition for EZH2 with a Ki value of 3 nM. EPZ-011989 trifluoroacetate shows robust methyl mark inhibition and anti-tumor activity. EPZ-011989 trifluoroacetate can be used for the research of various cancers. EPZ011989 trifluoroacetate is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition CuAAc with molecules containing Azide groups.

