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Falnidamol
GENERAL CATALOGUE

Falnidamol

HY-10322 · Free Sample (0.1 - 0.2 mg)

MedChemExpress · Cat: HY-10322

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medchemexpress.com/BIBX-1382.html
Catalog No: HY-10322
CAS No: 196612-93-8
Category: JAK STAT Signaling
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress

Description

Falnidamol BIBX 1382 is an orally active, selective EGFR tyrosine kinase inhibitor with an IC50 of 3 nM. Falnidamol displays > 1000-fold lower potency against ErbB2 IC50=3.4 ?M and a range of other related tyrosine kinases IC50 10 ?M. Falnidamol is a pyrimido-pyrimidine compound and has anti-cancer activity.

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