

HY-10409R · 5 mg
MedChemExpress · Cat: HY-10409R
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medchemexpress.com/fedratinib-standard.htmlDescription
Fedratinib Standard is the analytical standard of Fedratinib. This product is intended for research and analytical applications. Fedratinib TG-101348 is a potent, selective, ATP-competitive and orally active JAK2 inhibitor with IC50s of 3 nM for both JAK2 and JAK2V617F kinase. Fedratinib shows 35- and 334-fold selectivity over JAK1 and JAK3, respectively. Fedratinib induces cancer cell apoptosis and has the potential for myeloproliferative disorders research.







