

HY-144896 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-144896
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Manufacturer product page
medchemexpress.com/fht-1015.html
Description
FHT-1015 is a selective SMARCA4 IC50 = 4 nM and SMARCA2 IC50 = 5 nM also known as BRG1 and BRM inhibitor. FH-1015 is an allosteric inhibitor that causes conformation change in the BRG1/BRM protein upon interaction with an allosteric site, inhibiting ATPase activity. FH-1015 interferes with tumor cell growth and migration. FH-1015 can be studied in research for uveal melanoma and hematologic cancer.

