

HY-15791 · 50 mg
MedChemExpress · Cat: HY-15791
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medchemexpress.com/fr173657.htmlDescription
FR173657 is an orally active bradykinin B2 receptor antagonist IC50: 0.56, 1.5, 2.9 nM for pig, rat, human B2 receptor respectively . FR173657 p.o. inhibits BK-induced bronchoconstriction in guinea-pigs ED50: 0.075 mg/kg . FR173657 p.o. also inhibits Carrageenin-induced paw oedema in mice ED50: 6.8 mg/kg . FR173657 can be used for research of inflammatory disease.







