

HY-142941 · 50 mg
MedChemExpress · Cat: HY-142941
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medchemexpress.com/glucocorticoid-receptor-in-1.htmlDescription
Glucocorticoid receptor-IN-1 Compound WX002 is a selective glucocorticoid receptor GR modulator with anti-inflammatory effect. Glucocorticoid receptor-IN-1 exhibits very good transcriptional repressive activity with an IC50 of 2.11 nM against hMMP1, and transcriptional activation activity with an EC50 of 5.59 nM against MMTV.







