

HY-142942 · 50 mg
MedChemExpress · Cat: HY-142942
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medchemexpress.com/glucocorticoid-receptor-in-2.htmlDescription
Glucocorticoid receptor-IN-2 Compound WX019 is a selective glucocorticoid receptor GR modulator with anti-inflammatory effect. Glucocorticoid receptor-IN-2 exhibits very good transcriptional repressive activity with an IC50 of 0.171 nM against hMMP1, and comparable transcriptional activation activity with an EC50 of 0.94 nM against MMTV.







