

HY-163673 · 50 mg
MedChemExpress · Cat: HY-163673
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medchemexpress.com/glucocorticoid-receptor-modulator-4.html...Description
Glucocorticoid receptor modulator 4 Compound DL5 is a conjugate of a linker and a glucocorticoid receptor modulator. Glucocorticoid receptor modulator 4 exhibits GRE Reporter activity in mTNF expressing K562 cell with an EC50 of 40 ?M. Glucocorticoid receptor modulator 4 binds with an anti-tumor necrosis factor TNF antibody, and exhibits anti-inflammtory activity against arthritis in mouse models.