GENERAL CATALOGUE
GRPR antagonist-1
HY-115974 · 50 mg
MedChemExpress · Cat: HY-115974
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medchemexpress.com/grpr-antagonist-1.htmlCatalog No: HY-115974
CAS No: 3052544-28-9
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress
Description
GRPR antagonist-1 is a potent gastrin releasing peptide receptor GRPR antagonist, having the cytotoxicity against certain cancer cells IC50 of 4.97, 4.36 and 3.40 ?M in PC3, Pan02 and HGC-27 cells, respectively . GRPR antagonist-1 inhibits HGC-27 cell viability by decreasing the Bcl-2 level and increasing the Bax level, causing apoptosis, with anticancer activity.
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