

HY-136570 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-136570
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medchemexpress.com/gsk778.htmlDescription
GSK778 iBET-BD1 , a chemical probe, is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM BRD2 BD1 , 41 nM BRD3 BD1 , 41 nM BRD4 BD1 , and 143 nM BRDT BD1 , respectively. GSK778 phenocopies the effects of pan-BET inhibitors in cancer models.







