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GSK778 hydrochloride
GENERAL CATALOGUE

GSK778 hydrochloride

HY-136570A · 50 mg

MedChemExpress · Cat: HY-136570A

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Catalog No: HY-136570A
CAS No: 2863657-79-6
Category: Apoptosis
Pack Size: 50 mg
Brand: MedChemExpress

Description

GSK778 iBET-BD1 hydrochloride is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM BRD2 BD1 , 41 nM BRD3 BD1 , 41 nM BRD4 BD1 , and 143 nM BRDT BD1 , respectively.

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