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GENERAL CATALOGUE
GSK973
HY-138563 · 5 mg
MedChemExpress · Cat: HY-138563
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medchemexpress.com/gsk973.htmlCatalog No: HY-138563
CAS No: 2138473-38-6
Category: Epigenetics
Pack Size: 5 mg
Brand: MedChemExpress
Description
GSK973, a chemical probe, is a highly selective, orally bioavailable inhibitor of the BD2s second bromodomains of the BET family, with a pIC50 of 7.8 and a pKd of 8.7 for BRD4 BD2. GSK973 displays a 1600-fold selectivity for BRD4 BD2 over BRD4 BD1. GSK973 shows good potency against BRD2 BD2, BRD3 BD2, and BRDT BD2 pIC50=7.47.8; pKd=8.38.5 .