

HY-150684 · 50 mg
MedChemExpress · Cat: HY-150684
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/gxh-ii-052.htmlDescription
GXH-II-052 is a potent bivalent bromodomain and extraterminal domain BET inhibitor. GXH-II-052 shows binding potential for BRD4-1, BRD4-2, BRD4-T, BRDT-1, BRDT-2, BRDT-T with Kd values of 28, 9.1, 4.8, 0.6, 8.4, 2.6 nM, respectively. GXH-II-052 shows antiproliferative activity. GXH-II-052 decreases the expression of c-Myc.

