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HDAC8-IN-2
GENERAL CATALOGUE

HDAC8-IN-2

HY-144098 · 50 mg

MedChemExpress · Cat: HY-144098

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medchemexpress.com/hdac8-in-2.html
Catalog No: HY-144098
CAS No: 2824131-20-4
Category: Anti-infection
Pack Size: 50 mg
Brand: MedChemExpress

Description

HDAC8-IN-2 compound 5o is a potent HDAC8 inhibitor, with IC50 values of 0.27 and 0.32 ?M for smHDAC8 Schistosoma mansoni histone deacetylase 8 and hHDAC8, respectively. HDAC8-IN-2 shows significant killing of the schistosome larvae. HDAC8-IN-2 markedly impairs egg laying of adult worm pairs.

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