

HY-19760 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-19760
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medchemexpress.com/BET-IN-1.htmlDescription
I-BET282 is a pan-inhibitor of all eight BET bromodomains, and selectivity over other representative bromodomain-containing proteins. I-BET282 shows pIC50s ranging 6.4-7.7 for BRD2 BD1/BD2 , BRD2 BD1/BD , BRD3 BD1/BD , and BRD4 BD1/BD .