

HY-19826 · 50 mg
MedChemExpress · Cat: HY-19826
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Manufacturer product page
medchemexpress.com/isofistularin-3.html
Description
Isofistularin-3 is a direct, DNA-competitive DNMT1 inhibitor, with an IC50 of 13.5 ?M. Isofistularin-3, as a DNA demethylating agent, induces cell cycle arrest and sensitization to TRAIL in cancer cells. Isofistularin-3 can be used as an ADC cytotoxin.







