BioMall
KOR agonist 1
GENERAL CATALOGUE

KOR agonist 1

HY-161539 · 50 mg

MedChemExpress · Cat: HY-161539

Reach 3+ verified distributors

Manufacturer product page

medchemexpress.com/kor-agonist-1.html
Catalog No: HY-161539
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress

Description

KOR agonist 1 Compound 7a is a selective agonist for opioid receptor, with EC50s of 3.4, 701.2 and 1649 nM, for KOR, MOR and DOR, respectively. KOR agonist 1 binds KOR, MOR and DOR, with Kis of 3.9, 1053 and 4196 nM, respectively. KOR agonist 1 exhibits antinociceptive effect in ICR mouse model ED50 in hot plate test is 0.3 mg/kg, in abdominal constriction test is 0.2 mg/kg .

More from MedChemExpress

GPR120 Agonist 1
GPR120 Agonist 1
HY-108711
GPCR G Protein
AG-045572
AG-045572
HY-107534
GPCR G Protein
Pamabrom
Pamabrom
HY-17391
GPCR G Protein
ZD-7114
ZD-7114
HY-101320
GPCR G Protein
Vasopressin Dimer (anti-parallel) (TFA)
Vasopressin Dimer (anti-parallel) (TFA)
HY-P5214
GPCR G Protein
Zimeldine-d6
Zimeldine-d6
HY-118835S
GPCR G Protein
ZM241385 (Standard)
ZM241385 (Standard)
HY-19532R
GPCR G Protein
(5S,6S)-DiHETE
(5S,6S)-DiHETE
HY-130138
GPCR G Protein