

HY-130622 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-130622
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/lt052.html
Description
LT052 is a highly selective BET BD1 inhibitor with an IC50 of 87.7 nM. LT052 exhibits nanomolar BRD4 BD1 potency and 138-fold selectivity over BRD4 BD2 IC50=12.130 ?M . LT052 has anti-inflammatory?activity and can be used for acute gout arthritis research.

