Lumateperone-CHC,d3 tosylate

Description

Lumateperone-13C,d3 ITI-007-13C,d3 tosylate is 13C and deuterium labeled Lumateperone tosylate . Lumateperone ITI-007 tosylate is a 5-HT2A receptor antagonist Ki = 0.54 nM , a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors Ki = 32 nM , and a dopamine D1 receptor modulator. Lumateperone tosylate has anticancer activity and can also be used in studies of psychiatric disorders such as schizophrenia.