

HY-124069 · 50 mg
MedChemExpress · Cat: HY-124069
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Manufacturer product page
medchemexpress.com/m-525.html
Description
M-525 is a first-in-class, highly potent, irreversible and covalent menin-MLL protein-protein interaction inhibitor. M-525 binds to menin with an IC50 of 3 nM and achieves low nanomolar potencies in cell growth inhibition and in suppression of MLL regulated gene expression in MLL leukemia cells. Anti-leukemia activity.

