

HY-159177 · 50 mg
MedChemExpress · Cat: HY-159177
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/m4-machr-modulator-1.htmlDescription
M4 mAChR Modulator-1 compound 23i is a M4 mAChR positive allosteric modulator PAM . M4 mAChR Modulator-1 exhibits significantly greater cooperativity with ACh in ?-arrestin recruitment over G protein activation. M4 mAChR Modulator-1 displays weak PAM effect in G protein-mediated responses, but strong PAM effect in ?-arrestin recruitment.







