

HY-B0678S · 1 mg
MedChemExpress · Cat: HY-B0678S
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Manufacturer product page
medchemexpress.com/metaxalone-d3.html
Description
Metaxalone-d3 is the deuterium labeled Metaxalone. Metaxalone AHR438; NSC170959 is an FDA-approved muscle relaxant. Metaxalone acts mainly on the central nervous system and achieves muscle relaxation by inhibiting polysynaptic reflex arcs. In addition, Metaxalone is an inhibitor of MAO-A, which has anti-inflammatory and antioxidant effects. Metaxalone inhibits IL-1?-induced inflammatory phenotype, modulates NF-?B and other related signaling pathways, and decreases MAO-A expression and activity in IL-1?-treated microglia.