

HY-B0678 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-B0678
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medchemexpress.com/Metaxalone.htmlDescription
Metaxalone AHR438; NSC170959 is an FDA-approved muscle relaxant. Metaxalone acts mainly on the central nervous system and achieves muscle relaxation by inhibiting polysynaptic reflex arcs. In addition, Metaxalone is an inhibitor of MAO-A, which has anti-inflammatory and antioxidant effects. Metaxalone inhibits IL-1?-induced inflammatory phenotype, modulates NF-?B and other related signaling pathways, and decreases MAO-A expression and activity in IL-1?-treated microglia.