GENERAL CATALOGUE
ML221
HY-103254 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-103254
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medchemexpress.com/ML221.html
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Catalog No: HY-103254
CAS No: 877636-42-5
Category: GPCR G Protein
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress
Description
ML221 is a potent apelin APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 ?M in the cAMP assay, and 1.75 ?M in the ?-arrestin assay, and EC80 of 10 nM in both assays.
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