GENERAL CATALOGUE
Mozavaptan
HY-18346 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-18346
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medchemexpress.com/Mozavaptan.htmlCatalog No: HY-18346
CAS No: 137975-06-5
Category: GPCR G Protein
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress
Description
Mozavaptan OPC-31260 is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan shows 85-fold selectivity for V2 receptor over V1 receptor IC50 of 1.2 ?M , and can antagonize the antidiuretic action of arginine vasopressin AVP in vivo. Mozavaptan has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone SIADH , and congestive heart failure treatment.
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