

HY-18346R · 5 mg
MedChemExpress · Cat: HY-18346R
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Manufacturer product page
medchemexpress.com/mozavaptan-standard.html
Description
Mozavaptan Standard is the analytical standard of Mozavaptan. This product is intended for research and analytical applications. Mozavaptan OPC-31260 is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan shows 85-fold selectivity for V2 receptor over V1 receptor IC50 of 1.2 ?M , and can antagonize the antidiuretic action of arginine vasopressin AVP in vivo. Mozavaptan has the potential for hyponatremia, syndrome of inappropriate antidiuretic hormone SIADH , and congestive heart failure treatment.