

HY-101308A · 1 mg
MedChemExpress · Cat: HY-101308A
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Manufacturer product page
medchemexpress.com/mrs2179-tetrasodium-hydrate.html
Description
MRS2179 tetrasodium hydrate is a competitive P2Y1 receptor antagonist, with a Kb of 102 nM and a pA2 of 6.99 for turkey P2Y1 receptor. MRS2179 tetrasodium hydrate is selective for P2Y1 over P2X1 IC50=1.15 AAasAasAAmuM , P2X3 12.9 AAasAasAAmuM , P2X2, P2X4, P2Y2, P2Y4, and P2Y6 receptors. MRS2179 tetrasodium hydrate inhibits platelet aggregation.







