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MRS2690 disodium
GENERAL CATALOGUE

MRS2690 disodium

HY-116295A · 50 mg

MedChemExpress · Cat: HY-116295A

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Catalog No: HY-116295A
Category: GPCR G Protein
Pack Size: 50 mg
Brand: MedChemExpress

Description

MRS2690 disodium is a selective P2Y14 receptor agonist. MRS2690 disodium inhibits adenylyl cyclase activity, thereby reducing intracellular cAMP levels and mediating concentration-dependent vasoconstriction of porcine coronary arteries. MRS2690 disodium induces intracellular calcium mobilization, activates P38 and stimulates 35S GTP?S binding to RBL-2H3 cell membranes. MRS2690 enhances antigen NP-BSA -, C3a-induced ?-hexosaminidase ?-Hex release. MRS2690 disodium can be used for ischemic heart disease.

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