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MRT00033659
GENERAL CATALOGUE

MRT00033659

HY-117857 · Free Sample (0.1 - 0.2 mg)

MedChemExpress · Cat: HY-117857

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medchemexpress.com/mrt00033659.html
Catalog No: HY-117857
CAS No: 1401731-54-1
Category: Apoptosis
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress

Description

MRT00033659 is a potent broad-spectrum kinase inhibitor of CK1 IC50=0.9 ?M for CK1? and CHK1 IC50=0.23 ?M . MRT00033659, a pyrazolo-pyridine analogue, induces p53 pathway activation and E2F-1 destabilisation.

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