

HY-120000 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-120000
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medchemexpress.com/ms402.htmlDescription
MS402 is a BD1-selective BET BrD inhibitor with Kis of 77 nM, 718 nM, 110 nM, 200 nM, 83 nM, and 240 nM for BRD4 BD1 , BRD4 BD2 , BRD3 BD1 , BRD3 BD2 , BRD2 BD1 and BRD2 BD2 , respectively. MS402 blocks Th17 cell differentiation and ameliorates colitis in mice.