GENERAL CATALOGUE
MS645
HY-125232 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-125232
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Catalog No: HY-125232
CAS No: 2250091-96-2
Category: Epigenetics
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress
Description
MS645 is a bivalent BET bromodomains BrD inhibitor with a Ki of 18.4 nM for BRD4-BD1/BD2. MS645 spatially constrains bivalent inhibition of BRD4 BrDs resulting in a sustained repression of BRD4 transcriptional activity in solid-tumor cells.