

HY-107425 · 1 mg
MedChemExpress · Cat: HY-107425
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/MZ_1.htmlDescription
MZ 1 is a PROTAC connected by ligands for von Hippel-Lindau and BRD4. MZ 1 potently and rapidly induces reversible, long-lasting, and selective removal of BRD4 over BRD2 and BRD3. Kds of 382/120, 119/115, and 307/228 nM for BRD4 BD1/2, BRD3 BD1/2, and BRD2 BD1/2, respectively. Pink: BRD4 BD1BD2 ligand HY-13030 ; Blue: VHL ligand HY-125845 ; Black: linker HY-140189 .

