GENERAL CATALOGUE
NAS-181 dimesylate
HY-103156 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-103156
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Manufacturer product page
medchemexpress.com/nas181.htmlCatalog No: HY-103156
CAS No: 1217474-40-2
Category: GPCR G Protein
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress
Description
NAS181 is a potent and selective antagonist of rat 5-HT1B receptor, with a Ki of 47 nM. NAS181 shows 13-fold selectivity for r5-HT1B over bovine 5-HT1B receptor Ki=630 nM . NAS181 increases the 5-HT turnover and the synaptic concentration of 5-HT by inhibiting terminal r5-HT1B autoreceptors.
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