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NMDAR/HDAC-IN-1
GENERAL CATALOGUE

NMDAR/HDAC-IN-1

HY-147873 · 50 mg

MedChemExpress · Cat: HY-147873

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Catalog No: HY-147873
Category: Cell Cycle DNA Damage
Pack Size: 50 mg
Brand: MedChemExpress

Description

NMDAR/HDAC-IN-1 Compound 9d is a dual NMDAR and HDAC inhibitor with a Ki of 0.59 ?M for NMDAR and IC50 values of 2.67, 8.00, 2.21, 0.18 and 0.62 ?M for HDAC1, HDAC2, HDAC3, HDAC6 and HDAC8, respectively. NMDAR/HDAC-IN-1 efficiently penetrates the blood brain barrier.

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