

HY-100064R · 50 mg
MedChemExpress · Cat: HY-100064R
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medchemexpress.com/o-desmethyl-gefitinib-standard.htmlDescription
O-Desmethyl gefitinib Standard is the analytical standard of O-Desmethyl gefitinib. This product is intended for research and analytical applications. O-Desmethyl gefitinib is an active metabolite of Gefitinib in human plasma. The formation of O-desmethyl gefitinib is dependent on CYP2D6 activity. O-desmethyl gefitinib inhibits EGFR with an IC50 of 36 nM in subcellular assays.