

HY-129491 · 1 mg
MedChemExpress · Cat: HY-129491
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medchemexpress.com/o-desmethyl-pkc412.htmlDescription
O-Desmethyl Midostaurin CGP62221; O-Desmethyl PKC412 is the active metabolite of Midostaurin HY-10230 via cytochrome P450 liver enzyme metabolism. O-Desmethyl Midostaurin can be used as an indicator for Midostaurin metabolism in vivo. Midostaurin is a multi-targeted protein kinase inhibitor with IC50 ranging from 22-500 nM.

