

HY-14541S2 · 1 mg
MedChemExpress · Cat: HY-14541S2
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Manufacturer product page
medchemexpress.com/olanzapine-d8.html
Description
Olanzapine-d8 is a deuterated labeled Olanzapine. Olanzapine LY170053 is a selective, orally active monoaminergic antagonist with high affinity binding to serotonin H1, 5HT2A/2C, 5HT3, 5HT6 Ki=7, 4, 11, 57, and 5 nM, respectively , dopamine D1-4 Ki=11 to 31 nM , muscarinic M1-5 Ki=1.9-25 nM , and adrenergic ?1 receptor Ki=19 nM . Olanzapine is an atypical antipsychotic.