

HY-109067A · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-109067A
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Manufacturer product page
medchemexpress.com/opiranserin-hydrochloride.html
Description
Opiranserin VVZ-149 hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 GlyT2 and serotonin receptor 2A 5HT2A , with IC50s of 0.86 and 1.3 ?M, respectively. Opiranserin hydrochloride shows antagonistic activity on rP2X3 IC50=0.87 ?M . Opiranserin hydrochloride is development as an injectable agent for the treatment of postoperative pain.







