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Osimertinib-d6
GENERAL CATALOGUE

Osimertinib-d6

HY-15772S · 1 mg

MedChemExpress · Cat: HY-15772S

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Catalog No: HY-15772S
CAS No: 1638281-44-3
Category: JAK STAT Signaling
Pack Size: 1 mg
Brand: MedChemExpress

Description

Osimertinib-d6 is a deuterium labeled osimertinib. Osimertinib is a covalent, orally active, irreversible, and mutant-selective EGFR inhibitor with an apparent IC50 of 12 nM against L858R and 1 nM against L858R/T790M. Osimertinib overcomes T790M-mediated resistance to EGFR inhibitors in lung cancer.

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