

HY-159835 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-159835
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medchemexpress.com/oveporexton.htmlDescription
Oveporexton TAK-861 is an orally active and selective orexin receptor 2 OX2R agonist with an EC50 of 2.5 nM. Oveporexton exhibits 3000-fold selectivity for OX2R over OX1R. Oveporexton can be used for the study of hypersomnia disorders including narcolepsy.







