

HY-133529 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-133529
Reach 3+ verified distributors
Manufacturer product page
medchemexpress.com/pa-8.htmlDescription
PA-8 is a potent, selective and orally active PACAP type I PAC1 receptor antagonist. PA-8 inhibits the phosphorylation of CREB induced by PACAP in PAC1-, but not VPAC1- or VPAC2-receptor. PA-8 also inhibits PACAP-induced cAMP elevation with an IC50 of 2 nM.







