

HY-N6778 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-N6778
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medchemexpress.com/paxilline.htmlDescription
Paxilline is an indole alkaloid mycotoxin derived from Penicillium paxilli, which effectively inhibits the BK channel through a channel-blocking mechanism. Paxilline also inhibits sarco/endoplasmic reticulum Ca2+-stimulated ATPase SERCA , with IC50 values ranging from 5 ?M to 50 ?M for different SERCA isoforms. Paxilline exhibits significant anticonvulsant and neuroprotective effects, as well as certain antioxidant activity.







