

HY-151538 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-151538
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medchemexpress.com/pbrm1-bd2-in-8.htmlDescription
PBRM1-BD2-IN-8 compound 34 is a potent PBRM1 Bromodomain inhibitor PBRM1-BD2 Kd=4.4 ?M, PBRM1-BD2 IC50=0.16 ?M; PBRM1-BD5 Kd=25 ?M . PBRM1-BD2-IN-8 shows anti-cancer activity.

