GENERAL CATALOGUE
PD176252
HY-103286 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-103286
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medchemexpress.com/PD176252.htmlCatalog No: HY-103286
CAS No: 204067-01-6
Category: GPCR G Protein
Pack Size: Free Sample (0.1 - 0.2 mg)
Brand: MedChemExpress
Description
PD176252 is a potent antagonist of neuromedin-B preferring BB1 and gastrin-releasing peptide-preferring BB2 receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; PD176252 is also an agonist of N-Formyl peptide receptor1/2 FPR1/FPR2 , with EC50s of 0.31 and 0.66 ?M in HL-60 cells.