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PF-04577806
GENERAL CATALOGUE

PF-04577806

HY-139467 · 50 mg

MedChemExpress · Cat: HY-139467

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Manufacturer product page

medchemexpress.com/pf-04577806.html
Catalog No: HY-139467
CAS No: 1072100-81-2
Category: Epigenetics
Pack Size: 50 mg
Brand: MedChemExpress

Description

PF-04577806 is a potent, selective and ATP competitive PKC inhibitor. PF-04577806 shows potent inhibitory activity towards PKC?, PKC?I, PKC?II, PKC?, and PKC? with IC50s of 2.4 nM, 8.1 nM, 6.9 nM, 45.9 nM, and 29.5 nM, respectively. PF-04577806 can reverse retinal vascular leakage in diabetic rats.

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