

HY-155232 · 5 mg
MedChemExpress · Cat: HY-155232
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Manufacturer product page
medchemexpress.com/pi3k%CE%B4-in-16.html
Description
PI3K?-IN-16 is a potent and selective PI3K? inhibitor with an IC50 value of 0.9 nM. PI3K?-IN-16 has a strong anti-proliferative effect on SU-DHL-6 cells, causing cell cycle arrest and inducing apoptosis. PI3K?-IN-16 tightly bins to PI3K? protein with a planar-shaped conformation. The kinase activity of PI3K?-IN-16 which is 378-fold over PI3K?, 412-fold over PI3K?, and 10-fold over PI3K?. PI3K?-IN-16 can be used for the study of hematologic malignancies.







