

HY-161615 · 5 mg
MedChemExpress · Cat: HY-161615
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medchemexpress.com/protac-atr-degrader-2.htmlDescription
PROTAC ATR degrader-2 Compound 8i is a PROTAC degrader for ATR, through of . PROTAC ATR degrader-2 degrades ATR in acute myeloid leukemia AML cells MV-4-11 and MOLM-13, with DC50 of 22.9 and 34.5 nM. APROTAC ATR degrader-2 induces apoptosis, inhibits proliferations of AML cells. PROTAC ATR degrader-2 exhibits good pharmacokinetics charachers and antitumor efficacy against AML in mouse model. Pink: ATR ligand HY-161616 ; Blue:E3 ligase ligand Lenalidomide HY-A0003 ; Black: linker







