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PROTAC BRM/BRG1 degrader-3
GENERAL CATALOGUE

PROTAC BRM/BRG1 degrader-3

HY-168251 · 50 mg

MedChemExpress · Cat: HY-168251

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Catalog No: HY-168251
CAS No: 2933125-05-2
Category: Epigenetics
Pack Size: 50 mg
Brand: MedChemExpress

Description

PROTAC BRM/BRG1 degrader-3 compound 304 is a PROTACs-based BRM/BRG1 degrader with a DC50 of less than 1 nM for BRM degradation in SW1573 cells and a DC50 of greater than 1 nM for BRG1 degradation in SW1573 cells. PROTAC BRM/BRG1 degrader-3 has anti-tumor activity and anti-proliferative activity against A549 cells IC50=0.6 nM . Structure Note: PINK, Target protein ligand HY-168252 ; Blue, E3 HY-168253 ; Black, linker HY-69260 .

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