BioMall
Brand Store/MedChemExpress/PROTAC EGFR degrader 10
PROTAC EGFR degrader 10
GENERAL CATALOGUE

PROTAC EGFR degrader 10

HY-161632 · 50 mg

MedChemExpress · Cat: HY-161632

Reach 3+ verified distributors

Catalog No: HY-161632
CAS No: 3034244-56-6
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

PROTAC EGFR degrader 10 Compound B56 is a PROTAC degrader for epidermal growth factor receptor EGFR , with DC50 100 nM. PROTAC EGFR degrader 10 binds CRBN-DDB1 with a Ki of 37 nM. PROTAC EGFR degrader 10 degrades EGFR, focal adhesion kinase FAK , and RSK1, inhibits the proliferation of BaF3 wild type and EGFR mutants, with IC50 <150 nM.

More from MedChemExpress

STAT6-IN-2
STAT6-IN-2
HY-153991
JAK STAT Signaling
EGFR-IN-115
EGFR-IN-115
HY-162602
JAK STAT Signaling
ErbB-2-binding peptide
ErbB-2-binding peptide
HY-P4082
JAK STAT Signaling
TX2-121-1
TX2-121-1
HY-118998
JAK STAT Signaling
AZ7550
AZ7550
HY-B0794
JAK STAT Signaling
EGFR-IN-38
EGFR-IN-38
HY-144055
JAK STAT Signaling
CCT365623 hydrochloride
CCT365623 hydrochloride
HY-124674A
JAK STAT Signaling
HER2-IN-20
HER2-IN-20
HY-163657
JAK STAT Signaling