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PROTAC EGFR degrader 12
GENERAL CATALOGUE

PROTAC EGFR degrader 12

HY-171958 · 50 mg

MedChemExpress · Cat: HY-171958

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Catalog No: HY-171958
CAS No: 2654821-05-1
Category: JAK STAT Signaling
Pack Size: 50 mg
Brand: MedChemExpress

Description

PROTAC EGFR degrader 12 example 1 is a PROTAC degrader targeting EGFR that can effectively degrade EGFR mutants, but has little effect on EGFR WT. PROTAC EGFR degrader 12 shows IC50s against EGFRL858R-T790M NCI-H1975 cells , EGFRL858R NCI-H3255 cells , and EGFRL858R-T790M-L797S NCI-H1975+CS cells of all <50 nM.

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